CYP1A1

cytochrome P450 family 1 subfamily A member 1

Pharmacogene

Summary

This gene, CYP1A1, encodes a member of the cytochrome P450 superfamily of enzymes. The cytochrome P450 proteins are monooxygenases which catalyze many reactions involved in drug metabolism and synthesis of cholesterol, steroids and other lipids. This protein localizes to the endoplasmic reticulum and its expression is induced by some polycyclic aromatic hydrocarbons (PAHs), some of which are found in cigarette smoke. The enzyme's endogenous substrate is unknown; however, it is able to metabolize some PAHs to carcinogenic intermediates. The gene has been associated with lung cancer risk. A related family member, CYP1A2, is located approximately 25 kb away from CYP1A1 on chromosome 15. Alternative splicing results in multiple transcript variants encoding distinct isoforms. [provided by RefSeq, Jan 2016]

Known Variants52 total

rsidPosition (GRCh37)AllelesClassClinVar
rs180003115:74,719,894A/G3 prime UTR variant
rs2839943015:74,720,553G/Cmissense variant
rs5624020115:74,720,599G/Amissense variantlikely benign
rs4127918815:74,720,638G/Amissense variantbenign
rs7254750915:74,720,685A/Tmissense variant
rs7254751015:74,720,752C/CAframeshift variant
rs76821214015:74,721,236G/Astop gained
rs5631365715:74,721,463C/Amissense variant
rs14307067715:74,722,914C/Gmissense variant
rs464690315:75,011,641A/Gdownstream gene variant
rs498688315:75,012,217T/C3 prime UTR variant
rs5634342415:75,012,837C/Abenign
rs4546059715:75,012,896G/Abenign
rs74922364115:75,012,913C/Tuncertain significance
rs2839942915:75,012,925C/Tbenign
rs133066698115:75,012,927C/Guncertain significance
rs250552309215:75,012,931A/Guncertain significance
rs104894315:75,012,985T/Cmissense variantbenign
rs179981415:75,012,987G/Tmissense variantbenign
rs14703323315:75,012,995G/Alikely benign
rs76342769215:75,013,012C/Guncertain significance
rs14519886615:75,013,051T/Clikely benign
rs77019178015:75,013,078G/Auncertain significance
rs137915695915:75,013,313A/Tuncertain significance
rs75052097715:75,013,344C/Tuncertain significance
rs100813114715:75,013,363A/Guncertain significance
rs134997743615:75,013,367G/Clikely benign
rs74850725315:75,013,394G/Cuncertain significance
rs156719581415:75,013,544G/Auncertain significance
rs77849482915:75,013,558G/Tuncertain significance
rs75329876115:75,013,642C/Tuncertain significance
rs250552592115:75,013,787G/Tuncertain significance
rs498713315:75,014,027A/Glikely benign
rs75581518915:75,014,033C/Tuncertain significance
rs15051499315:75,014,646T/Cuncertain significance
rs6174760515:75,014,727G/Abenign
rs206317851515:75,014,765C/Tuncertain significance
rs37385891615:75,014,766C/Tuncertain significance
rs57752324715:75,014,799G/Cuncertain significance
rs14045978515:75,014,884G/Tuncertain significance
rs250552901315:75,014,891T/Cuncertain significance
rs15042796015:75,014,920C/Tlikely benign
rs76334619315:75,015,062T/Cuncertain significance
rs74587998215:75,015,124G/Tlikely benign
rs4552893515:75,015,161C/Tlikely benign
rs1786109415:75,015,206A/Gbenign
rs57825106815:75,015,262C/Tlikely benign
rs464642215:75,015,305C/Tmissense variantbenign
rs464642115:75,016,192G/T
rs260634515:75,017,176C/Aintron variant
rs247089315:75,019,449C/Tupstream gene variant
rs247229715:75,027,880C/Tintergenic variant

Gene information from NCBI Gene. Variant classifications from ClinVar.