CYP2E1

cytochrome P450 family 2 subfamily E member 1

Pharmacogene

Summary

This gene encodes a member of the cytochrome P450 superfamily of enzymes. The cytochrome P450 proteins are monooxygenases which catalyze many reactions involved in drug metabolism and synthesis of cholesterol, steroids and other lipids. This protein localizes to the endoplasmic reticulum and is induced by ethanol, the diabetic state, and starvation. The enzyme metabolizes both endogenous substrates, such as ethanol, acetone, and acetal, as well as exogenous substrates including benzene, carbon tetrachloride, ethylene glycol, and nitrosamines which are premutagens found in cigarette smoke. Due to its many substrates, this enzyme may be involved in such varied processes as gluconeogenesis, hepatic cirrhosis, diabetes, and cancer. [provided by RefSeq, Jul 2008]

Known Variants53 total

rsidPosition (GRCh37)AllelesClassClinVar
rs381386510:135,339,244G/Cdownstream gene variant
rs381386710:135,339,605G/Cdownstream gene variantno classification for the single variant
rs203192010:135,339,845C/Tdownstream gene variantno classification for the single variant
rs207067210:135,340,548A/Gdownstream gene variant
rs207067310:135,340,567A/Tdownstream gene variant
rs641342010:135,340,829G/Tdownstream gene variant
rs36795773110:135,340,948C/Tuncertain significance
rs75937242310:135,341,026G/Auncertain significance
rs249409541910:135,341,035T/Clikely benign
rs14374621110:135,341,054A/Guncertain significance
rs37442641210:135,341,994C/Guncertain significance
rs7255971010:135,342,034G/Amissense variant
rs75697388010:135,342,039G/Auncertain significance
rs2837174010:135,342,101G/Abenign
rs76429627310:135,342,117C/Tuncertain significance
rs54385500510:135,342,118C/Tuncertain significance
rs91590610:135,343,738C/Tupstream gene variant
rs819277210:135,344,711T/Cupstream gene variant
rs37342767210:135,345,212T/Guncertain significance
rs20116779310:135,345,633C/Guncertain significance
rs641341910:135,345,675G/Tmissense variant
rs2837174310:135,345,752T/Cbenign
rs77255923210:135,345,764C/Tlikely benign
rs57715940110:135,345,777C/Tuncertain significance
rs1225705410:135,346,018A/Gupstream gene variant
rs4129942610:135,346,202A/Glikely benign
rs249410429910:135,346,274A/Guncertain significance
rs249410431010:135,346,281A/Guncertain significance
rs74826897810:135,346,326A/Glikely benign
rs76650100410:135,346,335G/Auncertain significance
rs91590810:135,346,959G/Aupstream gene variant
rs74997900610:135,347,279G/Auncertain significance
rs77116094810:135,347,305G/Auncertain significance
rs2837174610:135,347,343C/Abenign
rs91590910:135,347,397T/Csynonymous variantbenign
rs464697610:135,347,727A/Gintron variant
rs819277510:135,348,026G/T
rs641343210:135,348,544T/Aintron variantassociation
rs74353510:135,349,367G/Aintron variant
rs132914910:135,349,801T/Cintron variant
rs14634406510:135,350,643C/Gbenign
rs15051490510:135,350,648T/Guncertain significance
rs249411042210:135,350,654C/Guncertain significance
rs207067610:135,351,137G/T
rs5589764810:135,351,264G/Amissense variant
rs5965637810:135,351,285G/Clikely benign
rs251564110:135,351,362T/Gmissense variantbenign
rs224969410:135,352,153A/T
rs224969510:135,352,168T/Cintron variant
rs2896938710:135,352,356A/Tbenign
rs5598223110:135,352,437G/Alikely benign
rs248025610:135,352,514A/T
rs251564410:135,353,079A/Cdownstream gene variant

Gene information from NCBI Gene. Variant classifications from ClinVar.