VKORC1

vitamin K epoxide reductase complex subunit 1

Pharmacogene

Summary

This gene encodes the catalytic subunit of the vitamin K epoxide reductase complex, which is responsible for the reduction of inactive vitamin K 2,3-epoxide to active vitamin K in the endoplasmic reticulum membrane. Vitamin K is a required co-factor for carboxylation of glutamic acid residues by vitamin K-dependent gamma-carboxylase in blood-clotting enzymes. Allelic variation in this gene is associated with vitamin k-dependent clotting factors combined deficiency of 2, and increased resistance or sensitivity to warfarin, an inhibitor of vitamin K epoxide reductase. Pseudogenes of this gene are located on chromosomes 1 and X. Alternative splicing results in multiple transcript variants. [provided by RefSeq, Aug 2015]

Known Variants46 total

rsidPosition (GRCh37)AllelesClassClinVar
rs20107502416:31,099,000C/Tbenign
rs88605193216:31,102,210C/Tuncertain significance
rs14175351216:31,102,212C/Tlikely benign
rs205728410016:31,102,283A/Tuncertain significance
rs88605193316:31,102,310A/Guncertain significance
rs729416:31,102,321C/Tupstream gene variantdrug response
rs205728623016:31,102,445G/Cuncertain significance
rs205728667216:31,102,500A/Guncertain significance
rs10489454216:31,102,564A/Cmissense variantdrug response
rs77770781616:31,102,568C/Tuncertain significance
rs720074916:31,102,589G/Asynonymous variantbenign
rs75357010516:31,102,595C/Glikely benign
rs205728781016:31,102,605G/Cuncertain significance
rs7254752816:31,102,655G/Amissense variantpathogenic
rs235961216:31,103,796A/Gregulatory region variantdrug response
rs254412546616:31,104,173G/Auncertain significance
rs37010535016:31,104,175C/Tlikely benign
rs37119751716:31,104,185T/Cbenign
rs805089416:31,104,509C/Tlikely benign
rs20013341816:31,104,649T/Auncertain significance
rs20104434816:31,104,713T/Cbenign
rs14527377216:31,104,714G/Auncertain significance
rs254412662816:31,104,734C/Tuncertain significance
rs76654960916:31,104,752G/Alikely benign
rs993443816:31,104,878G/Aregulatory region variantpathogenic
rs6174224516:31,104,878G/Tmissensedrug response
rs7254752916:31,105,274C/Tmissenseconflicting classifications of pathogenicity
rs1770847216:31,105,353G/Aregulatory region variantbenign
rs288473716:31,105,554A/Cregulatory region variantdrug response
rs20151554516:31,105,867C/Auncertain significance
rs10489454116:31,105,879T/Cmissense variantpathogenic
rs10489454016:31,105,917A/Gmissense variantpathogenic
rs6174223316:31,105,922G/Alikely benign
rs205731520616:31,105,934G/Auncertain significance
rs77407825816:31,105,939C/Guncertain significance
rs10489453916:31,105,966C/Amissense variantpathogenic
rs75925820416:31,105,987G/Auncertain significance
rs77189190616:31,105,997C/Auncertain significance
rs99337194316:31,106,011C/Tuncertain significance
rs5589476416:31,106,015C/Auncertain significance
rs75289235916:31,106,037C/Guncertain significance
rs88604269916:31,106,048C/Tuncertain significance
rs74570736716:31,106,052A/Guncertain significance
rs75985259916:31,106,095C/Tuncertain significance
rs56973735516:31,106,210C/Guncertain significance
rs992323116:31,107,689C/Tregulatory region variantpathogenic

Gene information from NCBI Gene. Variant classifications from ClinVar.

VKORC1 — vitamin K epoxide reductase complex subunit 1 — genewizard.net