ABCG2

ATP binding cassette subfamily G member 2 (JR blood group)

Pharmacogene

Summary

The membrane-associated protein encoded by this gene is included in the superfamily of ATP-binding cassette (ABC) transporters. ABC proteins transport various molecules across extra- and intra-cellular membranes. ABC genes are divided into seven distinct subfamilies (ABC1, MDR/TAP, MRP, ALD, OABP, GCN20, White). This protein is a member of the White subfamily. Alternatively referred to as a breast cancer resistance protein, this protein functions as a xenobiotic transporter which may play a major role in multi-drug resistance. It likely serves as a cellular defense mechanism in response to mitoxantrone and anthracycline exposure. Significant expression of this protein has been observed in the placenta, which may suggest a potential role for this molecule in placenta tissue. Multiple transcript variants encoding different isoforms have been found for this gene. [provided by RefSeq, Apr 2012]

Known Variants72 total

rsidPosition (GRCh37)AllelesClassClinVar
rs27252684:89,010,983A/Gbenign
rs12326066134:89,013,393T/Cuncertain significance
rs24760455854:89,013,406A/Guncertain significance
rs7806128214:89,013,463C/Tuncertain significance
rs347835714:89,013,496C/Tmissense variant
rs24760565064:89,015,772G/Auncertain significance
rs22311644:89,015,857C/Tintron variant
rs456055364:89,018,670C/Tlikely benign
rs7454730624:89,018,685T/Auncertain significance
rs24760736594:89,018,711A/Guncertain significance
rs10020125634:89,018,717G/Cuncertain significance
rs22311564:89,020,427C/Aintron variant
rs1921690634:89,020,503A/Gmissense variant
rs24760835034:89,020,515G/Tuncertain significance
rs7473097674:89,022,439T/Cuncertain significance
rs1807247064:89,023,741C/Tintron variant
rs27252644:89,026,109T/Cbenign
rs27252634:89,026,428C/Abenign
rs11957382084:89,028,358C/Auncertain significance
rs24761211464:89,028,418T/Auncertain significance
rs26226284:89,029,252C/Abenign
rs5361158584:89,030,372G/A
rs26226214:89,030,920C/Gregulatory region variant
rs131204004:89,033,527T/Cintron variant
rs7632968464:89,034,471T/Cuncertain significance
rs24761514574:89,034,514A/Guncertain significance
rs1386061164:89,034,589C/Tlikely benign
rs13250140914:89,034,677C/Auncertain significance
rs13324773284:89,036,148A/Guncertain significance
rs7631075054:89,036,183G/Cuncertain significance
rs7743973024:89,036,185G/Tuncertain significance
rs14810124:89,039,082A/Gintron variant
rs7719074144:89,039,258T/Clikely benign
rs11655642754:89,039,300C/Tuncertain significance
rs3879068704:89,039,310pathogenic
rs7794829564:89,039,311A/Cuncertain significance
rs2019135944:89,039,337G/Tuncertain significance
rs2001904724:89,039,366G/Astop gainedaffects
rs1402076064:89,039,396G/Astop gainedassociation
rs1490275454:89,044,180G/A
rs1384093704:89,044,312A/Tintron variant
rs21999364:89,045,331A/Gintron variant
rs1414719654:89,046,202C/Tintron variant
rs22311434:89,052,199T/Aintron variant
rs5289229394:89,052,295G/Cuncertain significance
rs22311424:89,052,323G/Tmissensedrug response
rs1439234184:89,052,339C/Tlikely benign
rs725527134:89,052,957G/Astop gainedassociation
rs22311394:89,052,964G/Abenign
rs22311384:89,053,718T/Cbenign
rs341241894:89,053,790G/Abenign
rs41481554:89,054,667A/Gintron variant
rs177315384:89,055,379G/Aintron variant
rs41481534:89,056,715G/Aintron variant
rs41481524:89,060,909T/Cintron variant
rs24762867574:89,061,033A/Cuncertain significance
rs22311374:89,061,114C/Tmissense variantassociation
rs31140184:89,064,581A/G
rs68576004:89,066,075C/Tregulatory region variant
rs177317994:89,068,455G/C
rs27252424:89,069,527T/G
rs99991114:89,073,197A/Cbenign
rs26226044:89,078,924T/A
rs31140204:89,083,666T/G
rs117329364:89,090,615A/Gintron variant
rs100117964:89,090,877T/Cintron variant
rs608165764:89,097,087G/Tintron variant
rs27252434:89,097,309G/T
rs74422244:89,102,651G/T
rs76721944:89,126,647C/A
rs794826594:89,145,931C/Tupstream gene variant
rs68462564:89,154,111G/A

Gene information from NCBI Gene. Variant classifications from ClinVar.