GRK4

G protein-coupled receptor kinase 4

Pharmacogene

Summary

This gene encodes a member of the guanine nucleotide-binding protein (G protein)-coupled receptor kinase subfamily of the Ser/Thr protein kinase family. The protein phosphorylates the activated forms of G protein-coupled receptors thus initiating its deactivation. This gene has been linked to both genetic and acquired hypertension. Several transcript variants encoding different isoforms have been found for this gene. [provided by RefSeq, Nov 2013]

Known Variants48 total

rsidPosition (GRCh37)AllelesClassClinVar
rs737921144:2,976,504G/Aintron variant
rs1913612004:2,986,296C/Auncertain significance
rs24747700464:2,986,305A/Cuncertain significance
rs3720270804:2,990,498C/Tuncertain significance
rs29603064:2,990,499G/Amissense variant
rs1425483154:2,990,546A/Guncertain significance
rs9369111914:2,990,556T/Cuncertain significance
rs29958034:2,990,864C/G
rs1424785774:2,994,002A/Clikely benign
rs13401270734:2,994,003G/Auncertain significance
rs3687095154:3,006,026G/Tuncertain significance
rs7492487624:3,006,030C/Tuncertain significance
rs10243234:3,006,043C/Tmissense
rs1381007964:3,009,471A/Guncertain significance
rs24751470194:3,009,491C/Guncertain significance
rs1174781494:3,009,536C/Tbenign
rs1412827434:3,011,382G/Auncertain significance
rs455389344:3,011,386C/Guncertain significance
rs5720387874:3,015,421G/Auncertain significance
rs7755408414:3,015,458G/Tuncertain significance
rs24752706434:3,015,491G/Auncertain significance
rs7459893044:3,015,542A/Guncertain significance
rs716082514:3,017,462A/Gintron variant
rs2012712304:3,021,391A/Cuncertain significance
rs12610478064:3,021,402C/Guncertain significance
rs24753914914:3,021,449C/Tuncertain significance
rs7576567014:3,021,473G/Auncertain significance
rs1859676764:3,021,475C/Tbenign
rs13416503434:3,021,527G/Auncertain significance
rs1394289414:3,024,158A/Cuncertain significance
rs2004719754:3,029,659C/Tuncertain significance
rs24755398334:3,029,669C/Guncertain significance
rs17380472024:3,029,693G/Clikely benign
rs5613613794:3,029,718C/Tlikely benign
rs13247082454:3,030,933G/Auncertain significance
rs7595524784:3,031,086G/Auncertain significance
rs1447717804:3,031,129G/Auncertain significance
rs5319179794:3,034,128C/A
rs9334028184:3,037,170G/Auncertain significance
rs2002164534:3,037,225T/Cuncertain significance
rs13773597064:3,039,129T/Cuncertain significance
rs18010584:3,039,150T/Cmissense
rs7787213464:3,039,158G/Auncertain significance
rs24756995684:3,039,168T/Guncertain significance
rs9288065584:3,039,188T/Cuncertain significance
rs7712207064:3,039,197C/Tuncertain significance
rs7640693314:3,039,231A/Cuncertain significance
rs3772706144:3,042,317C/Tuncertain significance

Gene information from NCBI Gene. Variant classifications from ClinVar.